Formulary
Imatinib [Specialist drug]: Indications, Dosing, Side Effects and Interactions
Imatinib [Specialist drug] clinical drug profile including indications, dosing, side effects, cautions and interactions.
MedNext Academy | 3 min read
Imatinib [Specialist drug]: Indications, Dosing, Side Effects and Interactions
Imatinib [Specialist drug] clinical drug profile including indications, dosing, side effects, cautions and interactions.
Indications and dose
**Chronic myeloid leukaemia,Acute lymphoblastic leukaemia,Gastro-intestinal stromal tumours,Myelodysplastic/myeloproliferative diseases,Dermatofibrosarcoma protuberans,Hypereosinophilic syndrome,Chronic eosinophilic leukaemia**
- **Adult** (By Mouth): Specialist drug - access specialist resources for dosing information.
Side effects
For imatinib [Specialist drug] Common or very common Alopecia; anaemia; appetite abnormal; asthenia; bone marrow disorders; chills; constipation; cough; diarrhoea; dizziness; dry eye; dry mouth; dyspnoea; excessive tearing; eye inflammation; fever; fluid imbalance; flushing; gastrointestinal discomfort; gastrointestinal disorders; haemorrhage; headaches; insomnia; joint disorders; muscle complaints; nausea; neutropenia; oedema; pain; photosensitivity reaction; sensation abnormal; skin reactions; sweat changes; taste altered; thrombocytopenia; vision blurred; vomiting; weight changes Uncommon Anxiety; arrhythmias; ascites; breast abnormalities; broken nails; burping; chest pain; CNS haemorrhage; congestive heart failure; depression; drowsiness; dysphagia; electrolyte imbalance; eosinophilia; eye discomfort; gout; gynaecomastia; hearing loss; hepatic disorders; hyperbilirubinaemia; hyperglycaemia; hypertension; hyperuricaemia; hypotension; increased risk of infection; laryngeal pain; lymphadenopathy; lymphopenia; malaise; memory loss; menstrual cycle irregularities; nerve disorders; oral disorders; palpitations; pancreatitis; peripheral coldness; pulmonary oedema; Raynaud's phenomenon; renal impairment; renal pain; respiratory disorders; restless legs; scrotal oedema; sepsis; sexual dysfunction; syncope; thrombocytosis; tinnitus; tremor; urinary frequency increased; vertigo Rare or very rare Angina pectoris; angioedema; arthritis; cardiac arrest; cataract; confusion; glaucoma; haemolytic anaemia; haemorrhagic ovarian cyst; hepatic failure (including fatal cases); hypersensitivity vasculitis; inflammatory bowel disease; intracranial pressure increased; muscle weakness; myocardial infarction; myopathy; nail discolouration; pericardial disorders; pulmonary fibrosis; pulmonary hypertension; seizure; severe cutaneous adverse reactions (SCARs); thrombotic microangiopathy; tumour lysis syndrome Frequency not known Embolism and thrombosis; hepatitis B reactivation; interstitial lung disease; neoplasm complications; osteonecrosis; pericarditis
Medicinal forms
Clinical governance
**Author:** MedNext Clinical Team. **Clinical reviewer:** Dr Shameer Deen, MBBS, MS, MRCS. **Sources:** BNF, Indian Pharmacopoeia, CIMS India. **Correction:** Report errors at support@mednext.academy.
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