Formulary
Busulfan [Specialist drug]: Indications, Dosing, Side Effects and Interactions
Busulfan [Specialist drug] clinical drug profile including indications, dosing, side effects, cautions and interactions.
MedNext Academy | 3 min read
Busulfan [Specialist drug]: Indications, Dosing, Side Effects and Interactions
Busulfan [Specialist drug] clinical drug profile including indications, dosing, side effects, cautions and interactions.
Indications and dose
**Chronic myeloid leukaemia**
- **Adult** (By Mouth): Specialist drug - access specialist resources for dosing information.
**Conditioning treatment before haematopoietic progenitor cell transplantation**
- **Adult** (By Mouth, Or By Intravenous Infusion): Specialist drug - access specialist resources for dosing information.
Contraindications
For busulfan [Specialist drug] Acute porphyrias
Side effects
For busulfan [Specialist drug] General side-effects: Common or very common Alopecia; diarrhoea; hepatic disorders; interstitial lung disease; nausea; sinusoidal obstruction syndrome; skin reactions; thrombocytopenia; vomiting Uncommon Seizure Rare or very rare Cataract; eye disorders Specific side-effects: Common or very common With intravenous use Anaemia; anxiety; appetite decreased; arrhythmias; arthralgia; ascites; asthenia; asthma; cardiomegaly; chest pain; chills; confusion; constipation; cough; depression; dizziness; dyspnoea; dysuria; electrolyte imbalance; embolism and thrombosis; fever; gastrointestinal discomfort; gastrointestinal disorders; haemorrhage; headache; hiccups; hyperglycaemia; hypersensitivity; hypertension; hypoalbuminaemia; hypotension; increased risk of infection; insomnia; mucositis; myalgia; nervous system disorder; neutropenia; oedema; pain; pancytopenia; pericardial effusion; pericarditis; reactivation of infections; renal disorder; renal impairment; respiratory disorders; stomatitis; vasodilation; weight increased With oral use Amenorrhoea (may be reversible); azoospermia; bone marrow disorders; cardiac tamponade; delayed puberty; hyperbilirubinaemia; infertility male; leucopenia; leukaemia; menopausal symptoms; oral disorders; ovarian and fallopian tube disorders; testicular atrophy Uncommon With intravenous use Capillary leak syndrome; delirium; encephalopathy; hallucination; hypoxia; intracranial haemorrhage Rare or very rare With oral use Dry mouth; erythema nodosum; gynaecomastia; myasthenia gravis; radiation injury; Sjgren's syndrome Frequency not known With intravenous use Hypogonadism; ovarian failure; premature menopause; sepsis Side-effects, further information Lung toxicity Discontinue if lung toxicity develops. Secondary malignancy Use of busulfan is associated with an increased incidence of secondary malignancy.
Medicinal forms
Capsule,Tablet,Solution
Clinical governance
**Author:** MedNext Clinical Team. **Clinical reviewer:** Dr Shameer Deen, MBBS, MS, MRCS. **Sources:** BNF, Indian Pharmacopoeia, CIMS India. **Correction:** Report errors at support@mednext.academy.
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